Dose of inhaled steroids

Recommendations:


Statement: inhaled steroids are slightly but significantly more effective when used four times daily than when used twice daily and are more effective when used twice daily than when used once daily, though the differences in lung function are not large (I).

Comment:
Five studies have looked at the effectiveness of differing dosage frequencies for inhaled steroids. They are all small studies, four of them are negative studies that do not have a power calculation in them and are therefore at risk of Type II errors. The group recognised the importance of compliance with treatment, though this was not formally studied; in most patients twice daily dosing is acceptable.

Boyd et al. (1985) studied 36 patients in a double blind, crossover double dummy study comparing 100 micro g of beclomethasone four times daily with 200 micro g twice daily. There was no difference in five symptoms. Clinic measured peak flow was 19 litres better in the four times daily group. There was no power calculation in this study.

Stiksa and Glennow (1985) studied 20 patients in an open crossover study of budesonide 800 micro g once daily; budesonide 400 micro g twice daily; and beclomethasone 200 micro g four times daily. There was no significant deterioration when on the once daily dose of budesonide. There was no power calculation in this study.

Munch et al. (1982) studied 20 patients in a double blind crossover design taking beclomethasone 200 micro g twice daily versus 100 micro g four times daily. There was no significant difference in peak flow or symptoms. There was no power calculation in this study.

Gagnon et al. (1994) studied 42 patients in a randomised double blind, double dummy crossover study of beclomethasone 500 micro g twice daily versus 1000 micro g in the afternoon versus 1000 micro g immediately before bed. Lung function was slightly better on the twice daily dosing. There was no power calculation in this study.

Toogood et al. (1982) studied 34 subjects who took inhaled budesonide in a complicated single blind randomised study using a block design which allowed comparison of three different budesonide dosages (400, 800, 1600 micro g per day); two dosing schedules (all dosages in the morning or dosages split between morning and evening); and two dosing frequencies (twice daily or four times daily). The results showed that both peak flow and FEV1 increased significantly as budesonide dosage increased; that peak flow, but not FEV1, was better with four times daily dose frequency than twice daily (20 litres per minute); and that there was no significant difference between the dosing schedules.

References
Boyd, G., Abdallah, S. and Clark, R. (1985) Twice or four times daily beclomethasone dipropionate in mild stable asthma? Clinical Allergy 15:383-389.

Gagnon, M., Cote, J., Milot, J., Turcotte, H. and Boulet, L.P. (1994) Comparative safety and efficacy of single or twice daily administration of inhaled beclomethasone in moderate asthma. Chest 105:1732-1737.

Munch, E.P. Taudorf, E. and Weeke, B. (1982) Dose frequency in the treatment of asthmatics with inhaled topical steroid. European Journal of Respiratory Diseases 63 Suppl 12:143-145.

Stiksa, G. and Glennow, C. (1985) Once daily inhalation of budesonide in the treatment of chronic asthma. A clinical comparison. Annals of Allergy 5: 49-51.

Toogood, J.H., Baskerville, J.C., Jennings, B., Lefcoe, N.M. and Johansson, S.A. (1982) Influence of dosing frequency and schedule on the response of chronic asthmatics to the aerosol steroid, budesonide. Journal of Allergy and Clinical Immunology 70:388-298.

Recommendation:


Statement: symptom control is better at high compared to low doses of inhaled steroids (I).

Comment:
Only a surprisingly small number of studies were identified to support this widely held clinical view.

Toogood et al. (1982) studied 34 subjects who took inhaled budesonide in

a complicated single blind randomised study using a block design which

allowed comparison of three different budesonide dosages (400, 800, 1600 micro g per day); two dosing schedules (all dosages in the morning or dosages split between morning and evening); and two dosing frequencies (twice daily or four times daily). The results showed that both peak flow and FEV1 increased significantly as budesonide dosage increased; that peak flow, but not FEV1, was better with four times daily dose frequency than twice daily; and that there was no significant different between the dosing schedules.

Dahl et al. (1993) (as above) compared four different doses of fluticasone with one dose of belcomethasone in five parallel groups. They showed that fluticasone produced a dose dependent increase in peak flow rates and dose dependent decrease in symptoms.

References
Dahl, R., Lundback, B., Malo, J.L., Mazze, J.A., Nieminen, M.M., Saarelainen, P. and

Barnacle, H.A. (1993) Dose-ranging study of fluticasone propionate in adult patients with moderate asthma. International Study Group. Chest 104:1352-1358.

Toogood, J.H., Baskerville, J.C., Jennings, B., Lefcoe, N.M. and Johansson, S.A. (1982) Influence of dosing frequency and schedule on the response of chronic asthmatics to the aerosol steroid, budesonide. Journal of Allergy and Clinical Immunology 70:388-398.

Decreasing steroid dosage

Recommendation:

Statement: we identified no direct evidence on when to decrease the dose of inhaled steroids. One study indirectly suggested that some patients on inhaled steroids may be over-treated (III).

Wong et al. (1993) studied patients on high dose inhaled steroids and attempted to reduce the dose using either nedocromil or a placebo in a double blind parallel study. There was little evidence from objective measures that nedocromil was significantly better than placebo. It was more interesting that a lot of the subjects were able to reduce corticosteroid dose considerably in both arms of the study.

References
Wong, C.S., Cooper, S., Britton, J.R. and Tattersfield, A.E. (1993) Steroid sparing effect of nedocromil sodium in asthmatic patients on high doses of inhaled steroids. Clinical and Experimental Allergy 23:370-376.

Research questions
When should inhaled steroids be decreased?

Is it effective to double inhaled steroids during inter current illnesses?

How safe are inhaled steroids?

Other inhaled anti-inflammatory agents

Recommendation:

Statement: nedocromil is more effective as a first line anti-inflammatory agent than placebo though its effect is not large (I). It has a questionable effect as a second line anti-inflammatory drug (I).

Edwards and Stevens (1993) reported a meta-analysis of nedocromil. The analysis included all double blind, placebo controlled studies supplied and analysed by Fisons. The trials were analysed in five groups only two of which are relevant: group one where nedocromil or placebo was added to baseline treatment with bronchodilators alone (whether oral or inhaled is not stated); and group four where patients were inadequately controlled on inhaled corticosteroids and nedocromil or placebo was added. The analysis did not include any studies comparing the addition of nedocromil against the addition of inhaled steroids. It is not stated what dose of steroids patients in group four were taking.

The results were analysed in terms of daily dose delivered: 8 mg or 16 mg. The outcome variables considered were: symptoms (the sum of 0-4 scales for patient-perceived severity of asthma and cough, each for both day and night); frequency of use of inhaled bronchodilators; pulmonary function tests (the mean of twice daily PEFR, change in FEV1 from baseline to final visit); and patient opinion (the proportion of patients saying the treatment was very or moderately effective).

Group one data involved 1689 patients, group four 1103. All figures quoted in the results are group mean changes.

In group one severity scores were on average half a scale point better with nedocromil, cough score was 0.3 scale points better, PEFR was ten litres per minute better in the lower dose group only, FEV1 was 0.2 litres better, inhaled bronchodilator use was one puff a day better and patient opinion was 20% better.

In group four severity score was 0.25 scale points better in the high dose group only, cough score was not different from placebo, PEFR was eight litres per minute better in the higher dose group only, FEV1 was not different from placebo, inhaled bronchodilator use was not different from placebo, and patient opinion was 14% better.

Nedocromil as a second line drug

Comment:
Our search identified four placebo studies not included in the meta-analysis and one second line study after the time frame of the meta-analysis.

Placebo studies

Chatterjee et al. (1986) compared nedocromil 4 mg four times daily with placebo. Nedocromil was slightly better in terms of bronchodilator use at night and day time symptoms.

Cua-Lim et al. (1986) studied a group of 54 asthmatic patients; nedocromil produced more improvement in symptoms and peak flow readings than placebo.

Greco et al. (1986) studied 130 subjects taking 4 mg of nedocromil four times daily, 2 mg four times daily or placebo; very small benefit of higher dose demonstrated.

van As et al. (1986) compared placebo with nedocromil twice daily and nedocromil four times daily. There were minor benefits compared with placebo with both nedocromil regimes.

Wong et al. (1993) studied patients on high dose inhaled steroids and attempted to reduce the dose using either nedocromil or a placebo in a double blind parallel study. There was little evidence from objective measurement that nedocromil was significantly better than placebo.

Comparison studies

Bergmann et al. (1989) compared nedocromil with beclomethasone in a single blind parallel group study comparing placebo, nedocromil and beclomethasone 400 g daily. Both drugs were better than placebo. Where differences between nedocromil and beclomethasone were present, these tended to favour beclomethasone.

Boldy and Ayres (1993) studied 77 patients treated with either nedocromil 4 mg four times daily or sodium cromoglycate 10 mg four times daily (no placebo). There were no clinically significant differences; any slight difference seemed to favour cromoglycate.

References
Bergmann, K.C., Bauer, C.P. and Overlack, A.A. (1989) Placebo-controlled, blind comparison of nedocromil sodium and beclomethasone dipropionate in bronchial asthma. Current Medical Research and Opinion 11:533-542.

Boldy, D.A. and Ayres, J.G. (1993) Nedocromil sodium and sodium cromoglycate in patients aged over 50 years with asthma. Respiratory Medicine 87:517-523.

Chatterjee, P.C., Fyans, P.G. and Chatterjee, S.S., (1986) A trial comparing nedocromil sodium (tilade) and placebo in the management of perennial bronchial-asthma. European Journal of Respiratory Diseases 69 Suppl. 147:314-316.

Cua-Lim, F., Agbayani, B.F. and Lachica, D. (1986) A double-blind comparative trial of nedocromil sodium and placebo in the management of bronchial asthma in patients routinely using oral bronchodilators. European Journal of Respiratory Diseases 69 Suppl. 147:306-310.

Edwards, A.M. and Stevens, M.T. (1993). The clinical efficiency of inhaled nedocromil sodium (Tilade) in the treatment of asthma. European Respiratory Journal 6: 35-41.

Greco, D.B., Negreiros, E.B., Chaieb, J.A., Ferreiralima, P. and Croce, J. (1986) A multicenter double-blind group comparative trial of 2 dose levels of nedocromil sodium and placebo in the management of perennial extrinsic-asthma. European Journal of Respiratory Diseases 69:323-326.

van As, A., Chick, T.W., Bodman, S.F., Storms, W.W., Nathan, R.A., Selner, J.C., Koepke, J.W., Townley, R.G., Bewtra, A.K., Nair, N., et al. (1986) A group comparative study of the safety and efficacy of nedocromil sodium (Tilade) in reversible airways disease: a preliminary report. European Journal of Respiratory Diseases 69 Suppl. 147:143-148.

Wong, C.S., Cooper, S., Britton, J.R. and Tattersfield, A.E. (1993) Steroid sparing effect of nedocromil sodium in asthmatic patients on high doses of inhaled steroids. Clinical and Experimental Allergy 23:370-376.


Statement: sodium cromoglycate is effective delivered in either a metered dose inhaler or a spinhaler (I).

Blumenthal et al. (1988) showed that sodium cromoglycate works better than placebo and equally well with metered dose inhaler when compared with spinhaler.

References
Blumenthal, M.N., Selcow, J., Spector, S., Zeiger, R.S., and Mellon, M. (1988) A multi-center evaluation of the clinical benefits of cromolyn sodium aerosol by metered dose

inhaler in the treatment of asthma. Journal of Allergy and Clinical Immunology 81:681-687.